Library Design, Search Methods, and Applications of Fragment-Based Drug Design
Rachelle J. Bienstock (Eds.)
Content: Overview : fragment based drug design --
Designing and searching fragment libraries --
Validation of reaction vectors for de novo design --
Design and application of fragment libraries for protein crystallography --
Ligand-based virtual screening using Bayesian inference network --
A computational fragment approach by mining the protein data bank: library design and bioisosterism --
Computational screening : docking --
A fragment based docking engine : eHiTS --
Fragment-based high-throughput docking and library tailoring --
Leads from fragments : fragment growing and linking --
Fragment-based high-throughput docking and library tailoring --
Fragment-based drug discovery for diseases of the central nervous system.
Designing and searching fragment libraries --
Validation of reaction vectors for de novo design --
Design and application of fragment libraries for protein crystallography --
Ligand-based virtual screening using Bayesian inference network --
A computational fragment approach by mining the protein data bank: library design and bioisosterism --
Computational screening : docking --
A fragment based docking engine : eHiTS --
Fragment-based high-throughput docking and library tailoring --
Leads from fragments : fragment growing and linking --
Fragment-based high-throughput docking and library tailoring --
Fragment-based drug discovery for diseases of the central nervous system.
Kategoriler:
Yıl:
2011
Yayımcı:
American Chemical Society
Dil:
english
Sayfalar:
197
ISBN 10:
0841224935
ISBN 13:
9780841224933
Seriler:
ACS Symposium Series 1076
Dosya:
PDF, 8.84 MB
IPFS:
,
english, 2011